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Items where Author is "Mieczkowski, Adam"

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Number of items: 29.

Article

Bojarska, Joanna and Łyczko, Krzysztof and Mieczkowski, Adam (2024) Synthesis, Crystal Structure and Supramolecular Features of Novel 2,4-Diaminopyrimidine Salts. Crystals, 14 (2). p. 133. ISSN 2073-4352

Belykh, Andrei and Hawro, Izabela and Kolczynska-Matysiak, Katarzyna and Loza-Valdes, Angel and Mieczkowski, Adam and Sumara, Grzegorz (2024) Triazolo[4,5-d]pyrimidin-5-amines based ERK3 inhibitors fail to demonstrate selective effects on adipocyte function. Archives of Biochemistry and Biophysics, 751 . p. 109825. ISSN 00039861

Burchiellaro, Katherine and Mieczkowski, Adam (2023) Synthesis and applications of cyclonucleosides: an update (2010–2023). Molecular Diversity . ISSN 1381-1991 (print) 1573-501X (web)

Park, Seongmin and Kim, Mingeun and Lin, Yuxi and Hong, Mannkyu and Nam, Geewoo and Mieczkowski, Adam and Kardos, Jozsef and Lee, Young-Ho and Lim, Mi Hee (2023) Designing multi-target-directed flavonoids: a strategic approach to Alzheimer's disease. Chemical Science, 14 (35). pp. 9293-9305.

Macyszyn, Julia and Burmistrz, Michal and Mieczkowski, Adam and Wojciechowska, Monika and Trylska, Joanna (2023) Conjugates of Aminoglycosides with Stapled Peptides as a Way to Target Antibiotic-Resistant Bacteria. ACS Omega, 8 (21). pp. 19047-19056. ISSN 2470-1343

Speina, Elzbieta and Wilczek, Marcin and Mieczkowski, Adam (2023) Dimeric Benzodiazepines as Peptide Mimetics to Overcome p53-Dependent Drug Resistance of Tumors. Biomolecules, 13 (2). p. 291. ISSN 2218-273X

Bojarska, Joanna and Mieczkowski, Adam and Ziora, Zyta M. and Skwarczyński, Mariusz and Toth, Istvan and Shalash, Ahmed O. and Parang, Keykavous and El-Mowafi, Shaima A. and Eman, H. M. Mohammed and Elnagdy, Sherif and AlKhazindar, Maha and Wolf, Wojciech M. (2021) Cyclic Dipeptides: The Biological and Structural Landscape with Special Focus on the Anti-Cancer Proline-Based Scaffold. Biomolecules, 11 (10). p. 1515. ISSN 2218-273X

Bieszczad, Bartosz and Garbicz, Damian and Świtalska, Marta and Dudek, Marta K. and Warszycki, Dawid and Wietrzyk, Joanna and Grzesiuk, Elzbieta and Mieczkowski, Adam (2021) Improved HDAC Inhibition, Stronger Cytotoxic Effect and Higher Selectivity against Leukemias and Lymphomas of Novel, Tricyclic Vorinostat Analogues. Pharmaceuticals, 14 (9). p. 851. ISSN 1424-8247

Mieczkowski, Adam and Speina, Elzbieta and Trzybiński, Damian and Winiewska-Szajewska, Maria and Wińska, Patrycja and Borsuk, Ewelina and Podsiadla-Bialoskorska, M and Przygodzki, Tomasz and Drabikowski, Krzysztof and Stanczyk, Lidia and Zhukov, Igor and Watala, Cezary and Woźniak, Krzysztof (2021) Diketopiperazine-Based, Flexible Tadalafil Analogues: Synthesis, Crystal Structures and Biological Activity Profile. Molecules, 26 (4). p. 794. ISSN 1420-3049

Piłsyk, Sebastian and Mieczkowski, Adam and Golan, Maciej and Wawrzyniak, Agata and Kruszewska, Joanna S. (2020) Internalization of the Aspergillus nidulans AstA Transporter into Mitochondria Depends on Growth Conditions, and Affects ATP Levels and Sulfite Oxidase Activity. International Journal of Molecular Sciences, 21 (20). ISSN 1422-0067

Bieszczad, Bartosz and Garbicz, Damian and Trzybiński, Damian and Dudek, Marta K. and Woźniak, Krzysztof and Grzesiuk, Elzbieta and Mieczkowski, Adam (2020) Unsymmetrically-Substituted 5,12-dihydrodibenzo[b,f][1,4]diazocine-6,11-dione Scaffold—A Useful Tool for Bioactive Molecules Design. Molecules, 25 (12). p. 2855. ISSN 1420-3049

Bieszczad, Bartosz and Garbicz, Damian and Trzybiński, Damian and Mielecki, Damian and Woźniak, Krzysztof and Grzesiuk, Elzbieta and Mieczkowski, Adam (2020) Unsymmetrically Substituted Dibenzo[b,f][1,5]-diazocine-6,12(5H,11H)dione—A Convenient Scaffold for Bioactive Molecule Design. Molecules, 25 (4). p. 906. ISSN 1420-3049

Wojciechowska, Monika and Równicki, Marcin and Mieczkowski, Adam and Miszkiewicz, Joanna and Trylska, Joanna (2020) Antibacterial Peptide Nucleic Acids—Facts and Perspectives. Molecules, 25 (3). p. 559. ISSN 1420-3049

Pilżys, Tomasz and Marcinkowski, Michał and Kukwa, Wojciech and Garbicz, Damian and Dylewska, Małgorzata and Ferenc, Karolina and Mieczkowski, Adam and Kukwa, Wojciech and Migacz, Ewa and Wołosz, Dominika and Mielecki, Damian and Klungland, Arne and Piwowarski, Jan and Poznański, Jarosław and Grzesiuk, Elzbieta (2019) ALKBH overexpression in head and neck cancer: potential target for novel anticancer therapy. Scientific Reports, 9 (1). p. 13249. ISSN 2045-2322

Mieczkowski, Adam and Wińska, Patrycja and Kaczmarek, Marta and Mroczkowska, Magdalena and Garbicz, Damian and Pilżys, Tomasz and Marcinkowski, Michał and Piwowarski, Jan and Grzesiuk, Elzbieta (2018) 2′-Deoxy-2′-azidonucleoside analogs: synthesis and evaluation of antitumor and antimicrobial activity. Chemical Papers, 72 (4). pp. 981-990.

Kasperowicz, Sławomir and Czerwińska, Jolanta and Majchrzak, Bartosz and Tudek, Barbara and Mieczkowski, Adam (2018) 5-Methyl-3,8-di-(2-amino-4-bromophenyl)-4,9-dioxa-1,2,6,7-tetraaza-5λ5-phosphaspiro[4.4]nona-2,7-diene. Molbank, 2017 (1). M978. ISSN 1422-8599

Dziełak, Monika and Trzybiński, Damian and Czerwińska, Jolanta and Majchrzak, Bartosz and Tudek, Barbara and Woźniak, Krzysztof and Mieczkowski, Adam (2018) N-(4-Bromobenzyl)-2-(5,6-dimethyl-1H-benzo[d]imid-azol-2-yl)benzeneamine. Molbank, 2018 (1). M979. ISSN 1422-8599

Mieczkowski, Adam and Psurski, Mateusz and Bagiński, Maciej and Bieszczad, Bartosz and Mroczkowska, Magdalena and Wilczek, Marcin and Czajkowska, Joanna and Trzybiński, Damian and Woźniak, Krzysztof and Wietrzyk, Joanna (2018) Novel (S)-1,3,4,12a-tetrahydropyrazino[2,1-c][1,4]benzodiazepine-6,12(2H,11H)-dione derivatives: Selective inhibition of MV-4-11 biphenotypic B myelomonocytic leukemia cells’ growth is accompanied by reactive oxygen species overproduction and apoptosis. Bioorganic & Medicinal Chemistry Letters, 28 (4). pp. 618-625.

Szakiel, Anna and Grabarczyk, Anna and Pączkowski, Cezary and Mieczkowski, Adam (2017) Comparison of the profiles of non-glycosylated triterpenoids from leaves of plants of selected species of genus Dioscorea. Phytochemistry Letters, 20 . pp. 350-355.

Mieczkowski, Adam and Trzybiński, Damian and Wilczek, Marcin and Psurski, Mateusz and Bagiński, Maciej and Bieszczad, Bartosz and Mroczkowska, Magdalena and Woźniak, Krzysztof (2017) (S)-2-(4-Chlorobenzoyl)-1,2,3,4-tetrahydrobenzo[e]pyrazino[1,2-a][1,4]diazepine-6,12(11H,12aH)-dione—Synthesis and Crystallographic Studies. Molbank, 2017 (4). M964. ISSN 1422-8599

Mieczkowski, Adam and Bieszczad, Bartosz (2016) Recent advances in the synthesis and applications of oxazolo[5,4-d]pyrimidines (microreview). Chemistry of Heterocyclic Compounds, 52 (10). pp. 782-784.

Zolnierczyk, Jolanta D. and Olejniczak, Agnieszka B and Mieczkowski, Adam and Blonski, Jerzy Z. and Kilianska, Zofia M and Robak, Tadeusz and Leśnikowski, Zbigniew J (2016) In vitro antileukemic activity of novel adenosine derivatives bearing boron cluster modification. Bioorganic & Medicinal Chemistry, 24 (21). pp. 5076-5087. ISSN 0968-0896

Mieczkowski, Adam and Tomczyk, Ewelina and Makowska, Małgorzata and Nasulewicz-Goldeman, Adam and Gajda, Roman and Woźniak, Krzysztof and Wietrzyk, Joanna (2016) Synthesis and Investigation of Anti-tumor Properties of Novel, Bicyclic Furopyrimidine, Pyrrolopyrimidine and Pyrimidopyridazine Nucleoside Analogues. Synthesis, 48 (4). pp. 566-572. ISSN 0039-7881

Mieczkowski, Adam and Bazlekova, Milena and Bagiński, Maciej and Wójcik, Jacek and Winczura, Alicja and Miazga, Agnieszka and Ghahe, Somayeh Shahmoradi and Gajda, Roman and Woźniak, Krzysztof and Tudek, Barbara (2016) A mild and efficient approach to the 6H-oxazolo[3,2-f]pyrimidine-5,7-dione scaffold via unexpected rearrangement of 2,3-dihydropyrimido[6,1-b][1,5,3]dioxazepine-7,9(5H,8H)-diones:synthesis, crystallographic studies, and cytotoxic activity screening. Tetrahedron Letters, 57 (7). pp. 743-746. ISSN 0040-4039

Gajda, Roman and Bagiński, Maciej and Tomczyk, Ewelina and Mieczkowski, Adam and Woźniak, Krzysztof (2015) Constrained nucleoside analogues – crystal and molecular structure of 6,5’ - O-anhydrouridines fixed in the anti conformation. Journal of Molecular Structure, 1097 . pp. 199-206. ISSN 0022-2860

Mieczkowski, Adam and Makowska, Małgorzata and Sekuła, Justyna and Tomczyk, Ewelina and Zalewska, Ewa and Nasulewicz-Goldeman, Adam and Wietrzyk, Joanna (2015) Bicyclic cytarabine analogues: synthesis and investigation of antitumor properties of novel, 6-aryl- and 6-alkyl-3H-pyrrolo[2,3-d] pyrimidin-2(7H)-one arabinosides. Tetrahedron, 71 (44). pp. 8458-8461. ISSN 0040-4020

Book Section

Adamska-Bartlomiejczyk, Anna and Bednarska, Katarzyna and Bialek-Pietras, Magdalena and Kilianska, Zofia M and Mieczkowski, Adam and Olejniczak, Agnieszka B and Paradowska, Edyta and Studzinska, Miroslawa and Sulkowska, Zofia and Zolnierczyk, Jolanta D. and Leśnikowski, Zbigniew J (2018) Boron Cluster Modification with Antiviral, Anticancer, and Modulation of Purinergic Receptors' Activities Based on the Nucleoside Structure. In: Boron-Based Compounds Potential and Emerging Applications in Medicine. Wiley, pp. 20-34. ISBN 978-1-119-27555-8

Conference or Workshop Item

Pilżys, Tomasz and Kukwa, Wojciech and Marcinkowski, Michał and Garbicz, Damian and Mieczkowski, Adam and Dylewska, Małgorzata and Grzesiuk, Elzbieta (2017) New inhibitors of ALKBH dioxygenases overexpressed in neck and head cancer. In: 42nd FEBS Congress: From Molecules to Cells and Back, 10-14 September 2017, Jerusalem, Israel.

Puszko, Anna and Sosnowski, P and Pułka-Ziach, Karolina and Laskowska, A and Mieczkowski, Adam and Perret, G and Misicka, Aleksandra (2016) Antiangiogenic activity and plasma stability study of peptidomimetics containing unnatural proline analogs. In: 34th European Peptide Symposium, Leipzig (Germany), 4-9.08.2016.

This list was generated on Fri Apr 26 06:11:39 2024 CEST.